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Design and synthesis of 4-(α-hydroxymalonyl)phenylalanine as a new phosphotyrosyl mimetic and its use in growth factor receptor bound 2 src-homology 2 (Grb2 SH2) domain-binding peptidesKANG, Sang-Uk; WORTHY, Karen M; BINDU, Lakshman K et al.Journal of medicinal chemistry (Print). 2005, Vol 48, Num 16, pp 5369-5372, issn 0022-2623, 4 p.Article

α-Substituted N-(4 -tert-butylbenzyl ) -N'-[4 -(methylsulfonylamino )-benzyl]thiourea analogues as potent and stereospecific TRPV1 antagonistsCHUNG, Jae-Uk; SU YEON KIM; CHOI, Sun et al.Bioorganic & medicinal chemistry. 2007, Vol 15, Num 18, pp 6043-6053, issn 0968-0896, 11 p.Article

Analysis of structure-activity relationships for the 'A-region' of N-(4-t-butylbenzyl)-N'-[4-(methylsulfonylamino)benzyl]thiourea analogues as TRPV1 antagonistsLEE, Jeewoo; KANG, Sang-Uk; MIN, Kyung-Hoon et al.Bioorganic & medicinal chemistry letters (Print). 2005, Vol 15, Num 18, pp 4136-4142, issn 0960-894X, 7 p.Article

Synthesis of tripeptides as potent Yersinia protein tyrosine phosphatase inhibitorsLEE, Kyeong; BOOVANAHALLI, Shanthaveerappa K; JUNG JUN LEE et al.Bioorganic & medicinal chemistry letters (Print). 2005, Vol 15, Num 18, pp 4037-4042, issn 0960-894X, 6 p.Article

Examination of acylated 4-aminopiperidine-4-carboxylic acid residues in the phosphotyrosyl+1 position of grb2 SH2 domain-binding tripeptidesKANG, Sang-Uk; WON JUN CHOI; OISHI, Shinya et al.Journal of medicinal chemistry (Print). 2007, Vol 50, Num 8, pp 1978-1982, issn 0022-2623, 5 p.Article

N-4-Substituted-benzyl-N'-tert-butylbenzyl thioureas as vanilloid receptor ligands: investigation on the role of methanesulfonamido group in antagonistic activityPARK, Hyeung-Geun; CHOI, Ji-Yeon; JEEWOO LEE et al.Bioorganic & medicinal chemistry letters (Print). 2004, Vol 14, Num 3, pp 787-791, issn 0960-894X, 5 p.Article

N-(3-acyloxy-2-benzylpropyl)-N'-[4-(methylsulfonylamino)benzyl]thiourea analogues: Novel potent and high affinity antagonists and partial antagonists of the vanilloid receptorLEE, Jeewoo; LEE, Jiyoun; OH, Uhtaek et al.Journal of medicinal chemistry (Print). 2003, Vol 46, Num 14, pp 3116-3126, issn 0022-2623, 11 p.Article

Analysis of structure-activity relationships for the 'B-region' of N-(4-t-butylbenzyl)-N'-[4-(methylsulfonylamino)benzyl ]- thiourea analogues as TRPV1 antagonistsLEE, Jeewoo; JIN, Mi-Kyoung; KIM, Sung-Eun et al.Bioorganic & medicinal chemistry letters (Print). 2005, Vol 15, Num 18, pp 4143-4150, issn 0960-894X, 8 p.Article

Novel potent antagonists of transient receptor potential channel, vanilloid subfamily member. 1 Structure-activity relationship of 1,3-diarylalkyl thioureas possessing new vanilloid equivalentsSUH, Young-Ger; LEE, Yong-Sil; KIM, Hee-Doo et al.Journal of medicinal chemistry (Print). 2005, Vol 48, Num 18, pp 5823-5836, issn 0022-2623, 14 p.Article

Structure-activity relationships of simplified resiniferatoxin analogues with potent VR1 agonism elucidates an active conformation of RTX for VR1 bindingLEE, Jeewoo; SU YEON KIM; WELTER, Jacqueline D et al.Bioorganic & medicinal chemistry. 2004, Vol 12, Num 5, pp 1055-1069, issn 0968-0896, 15 p.Article

N-4-t-Butylbenzyl 2-(4-methylsulfonylaminophenyl) propanamide TRPV1 antagonists: Structure-activity relationships in the A-regionKIM, Yong Soo; KIL, Min-Jung; JIN HEE LEE et al.Bioorganic & medicinal chemistry. 2012, Vol 20, Num 1, pp 215-224, issn 0968-0896, 10 p.Article

Examination of phosphoryl-mimicking functionalities within a macrocyclic Grb2 SH2 domain-binding platformKANG, Sang-Uk; SHI, Zhen-Dan; WORTHY, Karen M et al.Journal of medicinal chemistry (Print). 2005, Vol 48, Num 12, pp 3945-3948, issn 0022-2623, 4 p.Article

Analysis of structure-activity relationships for the 'b-region' of N-(3-acyloxy-2-benzylpropyl)-N'-[4-(methylsulfonylamino)-benzyl]thiourea analogues as vanilloid receptor antagonists: discovery of an N-hydroxythiourea analogue with potent analgesic activityLEE, Jeewoo; KANG, Sang-Uk; HA, Hee-Jin et al.Bioorganic & medicinal chemistry letters (Print). 2004, Vol 14, Num 9, pp 2291-2297, issn 0960-894X, 7 p.Article

N-[4-(methylsulfonylamino)benzyl]thiourea analogues as vanilloid receptor antagonists : Analysis of structure-activity relationships for the 'C-region'JEEWOO LEE; KANG, Sang-Uk; BLUMBERG, Peter M et al.Bioorganic & medicinal chemistry. 2004, Vol 12, Num 2, pp 371-385, issn 0968-0896, 15 p.Article